CaafimaadkaDiyaarinta

Daawada "Roxithromycin": tilmaamaha loo isticmaalo, sharaxaad, analogs, dib u eegista

In bukaanka qaar ka mid ah qiyaasta qoray "Roxithromycin"? Tilmaamaha isticmaalka kiniinka la oran tilmaamay doonaa. Sidoo kale ka soo maqaalka aad baran doontaa sida badan oo daroogada this, haddii uu wax analogues, waa maxay xasaasiyooyinka iyo sababo.

Curiska, sharaxaad, foomka daroogada

Kiniiniga "Roxithromycin" daahan filim, waa cadaan iyo hareeraheeda iyo biconvex qaab xardhan "164".

Walaxda firfircoon ee daroogada waa roxithromycin. Intaa waxaa dheer, daroogada ayaa sidoo kale ka mid ah qaybaha kaabayaal sida giproloza, K30 povidone, poloxamer, milmahayn magnesium, silica Kolloidol, galleyda iyo Rusheyn kartaa.

Iyadoo la tixgelinayo daahan filim, waxa ku jira hypromellose, dextrose, tones propylene iyo titanium dioxide.

iibinta daroogada bixisey in baakad fin iyo kartoonada siday u kala horreeyaan.

Sifooyinka pharmacological kiniinno antibiyootig

Waa maxay saamaynta on daawada jirka "Roxithromycin"? Tilmaamaha loogu isticmaalo dalalka waa antibiotic ah semisynthetic, tirsan kooxda macrolides, taas oo uu leeyahay spectrum balaadhan oo ah waxqabad antibiotic.

medicament waxay leedahay tallaabo bacteriostatic. Waxaa xidhana in ay 50s ee subunit ribosomal, gaabis Avv borotiinka ribosome, hakiyo reaction transpeptidation iyo translocation, iyo sidoo kale hababka of lagala kulmo dhexeeya silsilad peptide iyo acids amino. saamayn noocan oo kale kor u Iscelin ee koritaanka iyo taranka bakteeriyada.

Antibiotic "Roxithromycin" si fiican oo dhakhso ah guskiisa galay unugyada, kaas oo hubinaya in ay awood ka dhanka ah wareer intracellular sare.

Pharmacokinetics daroogada

Halkee nuugista ee "Roxithromycin" daroogada? khubaro Guest sheegay in ka dib markii maamulka afka of medicament la nuugo ka soo mareenka caloosha iyo mindhicirka.

Kiniiniga deggan deegaanka acidic ee caloosha. Cuntada, daroogada iyada saacadood ka dib markii ¼ medicament u saameyn ah kuma laha ay nuugista.

Ka dib markii la helo ay fiirsashada daroogada ugu badnaan gaari kadib markii bar ilaa laba saacadood.

Isticmaalka daroogada ee 13 saacadood kula bareeg ah ilaaliyaan uruureen baahan yahay ee daroogada ee dhiigga inta lagu jiro maalinta.

Isgaarsiinta la borotiinada plasma waa 95,5%. Xaaladdan oo kale, daroogada sambabbada, prostate makrii iyo qumanka. Sidoo kale waxaa la helay in unugyada (macrophages) iyo dheecaannada jidhka kala duwan.

"Roxithromycin", qiimaha kaas oo hoos ku qoran, ficil ahaan ma geli caqabad dhiig-maskaxda iyo saxarrada la caanaha naaska oo kaliya in tiro yar. Iyadoo ay taasi jirto, qaadan daroogada this xilliyada sida waa ka mamnuuc.

Daawada waxaa qayb ahaan metabolized beerka. Its saamiga ugu weyn (50%) waxaa raaca isbeddelin xiidmaha iyo dhex kelyaha (ku dhowaad 12%) iyo Nuur (qiyaastii 15%).

The bar-nolosha oo ah walaxda firfircoon ka dib markii dose hal waa qiyaastii 13 saacadood.

fiirsashada ugu badnaan iyo badh-nolosha ee kor u daroogada la beerka masaakiinta.

Tilmaamayaasha antibiotic

Waayo, waa maxay ujeedada qoray "Roxithromycin" kiniin? Tilmaamaha loogu isticmaalo dhigayaa in wakiilka this wax ku ool ah loogu daweeyo cudurada in waxa sababa wareer ah u nugul walaxda firfircoon.

daroogada Adult qoray waayo, nimankii aad:

  • qumanka, pharyngitis, hogaga ba'an;
  • cudurada unugyada jilicsan, iyo maqaarka,
  • pneumonia, boronkiitada,
  • cudurada kaadi mareenka,
  • cudurrada ilkaha (ilkaha iyo saabka afka).

"Roxithromycin" qoray ee carruurta:

  • pharyngitis, qumanka, hogaga ba'an;
  • pneumonia, boronkiitada,
  • cudurada unugyada jilicsan iyo maqaarka.

Sababo isticmaalka wakiilka antibiotic

Xaaladaha qaarkood, bukaanka ma qori daroogada "Roxithromycin"? Tilmaamaha loogu isticmaalo sida uu reebay soo socda:

  • dareenka kor u bukaan roxithromycin macrolides ama in oo dhan, iyo sidoo kale waxyaabaha kale ee dejinta;
  • porfyri;
  • inta aad uurka leedahay,
  • soo dhaweynta isku mar la "cisapride", "terfenadine," "pimozide" iyo "Astemizole";
  • miisaanka jidhka ka yar 40 kg,
  • naas-nuujinta,
  • wada jir ergot adag isticmaalka vasoconstrictive (kadeed iyo dihydroergotamine);
  • da'da 12 sano.

maamulka taxaddar of kiniiniyada

Drug "Roxithromycin", taas oo analogues la hoos ku soo bandhigi doonaa, si taxadir leh loo soo qoray in dadka qaba cagaarshowga ama kelyaha la'aan, bukaanada waayeelka ah, iyo dadka qaba xaaladaha in ay gacan xanuunada garaaca wadnaha, iyo Dheereyn dhasho xilliga QT ah.

qiyaasta of daroogada ee dadka waaweyn iyo carruurta

Kiniiniga gudaha qoray cuntada ka hor. Waayo, dadka waaweyn iyo carruurta ka weyn yahay 12 sano, qiyaasta caadiga ah waa 150 mg oo daroogada ah laba jeer maalintii dura 13 saacadood ama 300 mg dose (loogu talagalay dadka waaweyn).

Dadka waayeelka ah maalin walba iyo dhoos keli ah daawada aysan waxba ka beddelin. Bukaanka qaba daroogada la'aan kelyaha waxaa maamula ee dose oo ah 150 mg laba jeer maalintii.

Bukaanka qaba qiyaasta beerka waa la dhimay by badh (150 mg maalintii hal mar).

Muddada aad daawada ee dadka waaweyn iyo carruurta

Mudo intee leeg ayay qaadan doontaa daawada "Roxithromycin"? Muddada aad daawada ku xiran tahay calaamad muujinaysa, iyo sidoo kale noole ah oo keena cudurka, iyo adkaanta cudurka.

In dadka waaweyn, heerka caadiga ah qaadan kartaa oo ku saabsan 5-10 maalmood. In aan cudur waxaa keena streptococcus beta-hemolytic, therapy, waa in ugu yaraan 10 maalmood.

Iyadoo la tixgelinayo carruurta, muddada koorsada ay sidoo kale waa 5-10 maalmood.

medicament Overdosing

At qaadasho sare ee daawada bukaan kordhin kara waxyeelo dose-xiriira. Sida daaweynta xaaladaha sida isticmaalaya therapy astaamaha iyo lavage gastric.

waxyeellooyin

Iyadoo qaadashada tixgelinta daroogada ee bukaanka muujin karaan dhibaatooyinka soo socda:

  • lalabo, calool xanuun, matag, shuban, ulcerös pseudomembranous, ganaca,
  • kordhay dhaqdhaqaaqa of transaminases beerka, hepatocellular ba'an ama hepatitis cholestatic;
  • paraesthesia, dawakhaad, isbedel xagga dhadhanka, madax-xanuun, rabshooyin ee urta, lumis maqal waa ku meel gaar, dhalanteed, vertigo, Gipoakuzija;
  • casaan, finan, purpura;
  • anjioedema, bronchoconstriction, urtikaria, eosinophilia;
  • lama filaan ah anaphylactic, multiforme erythema ;
  • superinfection, candidiasis.

talooyin gaar ah

Dadka qaba daroogada beerka si taxadir leh xad-dhaaf ah u magacaabay.

Iyadoo horumarinta dareen diidmo oo xasaasiyadeed oo daawada superinfection waa in la joojiyo iyo bukaanka uu helo daaweyn sax ah.

Marka la helo daroogada, iyo sidoo kale laba ilaa saddex toddobaad ka dib daawaynta, bukaanka waxaa laga yaabaa in la horumariyo shuban sababa colitis pseudomembranous.

Drug "Roxithromycin" iyo khamriga waxaa ka mamnuuc ah in la isu geeyo.

isdhexgalka daroogada

daawo viewed aan la maamulo daawooyin ay ku jiraan kadeed ah, dihydroergotamine, ama, sida ay keeni kartaa dabac halbowlaha.

Ha qaadan "Roxithromycin" leh "terfenadine" sabab u ah kordhinta halista jahawareerka nidaamka wadnaha.

Wada jir ah ula gelitaanka ee daroogada la "digoxin" kordhin kartaa ay nuugista, taasoo keeni doonta in horumarka sarkhaan glycoside.

isku darka ah "Cyclosporine" ama "theophylline" with "Roxithromycin" keeni kordhin karaa uruureen plasma doonana.

medicament Analogs

The analoogga ugu caansan "Roxithromycin" waa "erythromycin". Guide dhigayaa in diyaarinta this sidoo kale waa antibiotic ah.

Sidaas oo ka mid ah qalabka fiican? Marka la barbar dhigo "erythromycin" "Roxithromycin" wuxuu leeyahay sifooyin pharmacokinetic more wanaagsanaaday. Ka dib markii maamulka afka, waxaa arrin si degdeg ah nuugo ka soo mareenka caloosha iyo mindhicirka.

Iyada oo bioavailability sare oo dheeraad ah, taas oo kullanka ku xidhan qaadashada cuntada, daawada la ogaado in dhiigga horay on saacadood ¼ ka dib.

Waa in sidoo kale la sheegay in ay daroogada "Roxithromycin" foomamka fiirsashada badan oo la taaban karo oo lagu kalsoonaan karo, ma aha oo kaliya in dheecaannada jidhka iyo unugyada, laakiin sidoo kale in serum dhiigga.

Sidaas darteed, waxaa si ammaan ah in la xuso karo in daawada ugu horeeyay ee labaad ka qaniintay ka xun. "Erythromycin", oo edbinta waxaa sidoo kale gundhig in kartoon ah, waa antibiotic huriye.

Intaa waxaa dheer ku yidhi hab, daroogada "Roxithromycin" waxaa lagu beddeli karaa oo daawooyin sida "Brilid", "Esparoksi" "Vero Roxithromycin", "Elroks", "Ksitrotsin", "Rusbrikar", "Remora", "Rulitsin", " Rokseptin "," Rulid "," RoksiGEKSAL "," Romik, "" Roksid "," Roksolit "," Roksilor "" Roxithromycin DS "," Roksimizan ".

daawo Price

Waa imisa antibiotic ah "Roxithromycin"? Qiimaha daroogada tani waa mid qaali ah. iibso farmasiyada noqon kartaa 550-600 rubles.

Kurtumm ku saabsan daawada

Antibiotic "Roxithromycin" - daroogada quruxsan caansan ka mid ah bukaanka. Sidaa darteed, waxaa jira tiro ka mid ah faalooyin oo ku saabsan qalab this xad. Dadka intooda badan sheegeen in daawada u dhaqmo sida daawada aad u wax ku ool ah antibiotic. In lagu daro daawooyinka kale ayuu ku dagaalama cudurada kala duwan ee mareenka sare iyo hoose ee neefsashada (qumanka, pharyngitis, hogaga ba'an), iyo mareenka Fistula, unugyada jilicsan iyo maqaarka.

Oo ay la socoto jawaab-celin wanaagsan ka qalab this la heli karo iyo taban. Inta badan, ee la soo dhaafay la xiriira waxyeelo ka dhaca bukaanlayda qaadato daawada hoos tixgelin. Bukaanjiifka qaar ayaa ka cabanaya lallabo, shuban daran, madax-xanuun, matag, xaalad xumeyd pankreatit iyo finan.

Marka aad aragto calaamadahan, dhakhaatiirta ku talinaynaa in ay diidaan in ay aqbalaan kiniin oo la arko dhakhtar, kuwaas waxaa waajib ku ah in ay talo daroogada ammaan ah.

Sidoo kale waa in la ogaadaa in ay jiraan wax badan oo dib u eegista in daroogada ayaa kharash buunbuuniyo. Bukaan-socodka sheegan in analogues of taasi ka dhigan tahay waxaa jira wax badan oo ka raqiisan iyo halka aan xad liita inuu waxtarka.

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