CaafimaadkaDiyaarinta

Daroogada Cardioselective "Metoprolol": tilmaamaha loo isticmaalo

The daroogada tilmaamaha "Metoprolol" loo isticmaalo waxaa loola jeedaa koox ka mid ah cardioselective beta-blockers in ay leeyihiin antiarrhythmic, antianginal iyo antihypertensive saamayn. daroogada Tani waxay u ogolaaneysaa for dib u dhac waqti gaaban ee tabinta AV ah, yareeyo automaticity ee sanka Guntin, contractility myocardial iyo excitability iyo in la yareeyo xaddiga garaaca wadnaha, wax soo saarka wadnaha iyo myocardial oksajiinta. Intaa waxaa dheer, daroogada cardioselective "Metoprolol", qiimaha taas oo ku saabsan shan iyo toban - labaatan rubles, wax ku ool ah uu hakiyo saamaynta stimulatory catecholamines on wadnaha la stress psycho-niyadeed iyo jidheed. Sida sifooyinka ugu muhiimsan ee pharmacokinetic daroogada, ay fiirsashada ugu badan ee plasma bilaabo inuu la calaamadeeyay ku saabsan mid ka mid ah ka dib markii - laba saacadood, iyo celceliska bar-nolosha ee loo yaqaan saddex ilaa toddoba saacadood.

Soo saaray daroogada hypotensive "metoprolol" (diiwaanka waxaa had iyo jeer ka mid ah) ee foomka of kaabsal wareega midabka cad-cream iyo foomka of xal loogu tala galay maamulka xididka xiga. Halabuurka The of this daroogada cardioselective sida qayb firfircoon waxaa ka mid tartrate metoprolol. Kiniiniga dheeraad ah ka kooban laktosmonohydrat lactose, cellulose mikrokristallin, povidone, milmahayn calcium, crospovidone iyo Rusheyn kartaa.

Isticmaal tilmaamaha antianginal iyo antiarrhythmic "Metoprolol" loo isticmaalo bixiya saaraha talinaysaa oo lagu daweeyo bukaanada qaba angina (oo ay ku jiraan post-Wadnaxanuun), hypertension iyo garaaca (oo ay ku jiraan nooca tachyarrhythmia supraventricular). Intaa waxaa dheer, arrin inta badan, dhakhaatiirta qoro dawooyinka hypotensive si looga hortago weerarrada dhanjafka. In daaweynta isku dhafan ee tayroodh waxa ay sidoo kale waxaa lagu talinayaa in la bilaabo qaata lacagaha cardioselective "Metoprolol". Tilmaamayaasha loogu tala galay in ka mid ah daawaynta dayactirka labada dib markii Wadnaxanuun myocardial. In daawada this kiis kasta oo shakhsi ah dhakhtar oo dhigaya keliya ku salaysan falanqayn kuwan.

Sida liiska sababo weyn daroogada oo ay jidhkiisa cardioselective waa horrayn lagama maarmaan ah in loo qoondeeyo dareen dheeraad ah si ay u tartrate metoprolol, iyo dareen-celinta xasaasiyad kasta qaybaha qofka jirran. Dadka qaba wadnaha, xannibaad atrioventricular, daran sanka bradycardia ama block sinoatrial la mid ah waa in aysan qaadan wax daawo ah oo antiarrhythmic "Metoprolol". Tilmaamaha loogu isticmaalo ayaa sidoo kale aan lagu talinayaa in this wakiilka antihypertensive la sanka buka, xanuunada wareegga dhiigga durugsan ee nidaamka ama hypotension. Iyada oo taxaddar dheeraad ah waa in la isticmaalo dawadan lacala tayroodh, mellitus sonkorowga, neefta, pheochromocytoma, hypoglycemia, daweeyay gravis, emphysema, psoriasis, aysiidh dheefshiidka, boronkiitada non-xasaasiyad ama niyadjabka.

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