Caafimaadka, Diyaarinta
Tilmaamaha loogu isticmaalo "tiapridal". Analogs iyo dib u eegis
"Tiapridal" - daawo waallida dajiya macmalay by tiapride. Daawada waxaa laga codsadaa sida ku dejinaysaa, xanuunka iyo hypnotic. Basis of tallaabo waallida dajiya - xanibeen receptors dopamine, taas oo si weyn u saameeya hawlaha yimaada habdhiska dhimirka. In this article waxaan ku tilmaami si faahfaahsan oo ku saabsan daroogada.
Qaab dhismeedka kooban daroogada
Daawada waxaa laga heli karaa laba nooc, kiniinka laga iibsan karaa oo xal:
- Mid ka mid ah kiniin sida mid dhalada ka kooban yahay 100 milligram ee ka kooban ugu weyn iyo walxaha kaabayaal ah. Sida maaddooyinka kaabayaal ah loo isticmaalo ee halabuurka ah ee povidone, milmahayn magnesium, mannitol. Halabuurka waxa kale oo kaabaya la dioxide Kolloidol, Silicon iyo mikrokristallin cellulosa ah aqueous.
- ka qayb ugu weyn ee xalka reebo kooban chloride sodium iyo biyo la isku duro.
In hal sanduuq oo ku jira 20 kaniini oo (2 finan 10 kiniin) ama 12 fijaan (2 finan of 6 fijaan). Tilmaamaha loogu isticmaalo "Tiapridal" ee foomka of xal la isku duro u ogolaanaya intravenously iyo intramuscularly maamulo. Qaabkan daroogada waa oo kaliya ku haboon oo lagu daweeyo bukaanada qaangaarka ah.
Pharmacodynamics "tiapridal"
medicament waxay leedahay neuroleptic, xanuunka iyo ficil anxiolytic. Sida Buugga edbinta, "Tiapridal" eegista blocks hawlaha of D 2 receptors ah dopamine dhexe. Sayidka on D 1 receptors saameyn ah kuma laha. daroogada uu uga takhalusi psoriasis, marka loo isticmaalo in dadka waayeelka ah hagaajinaysaa fekerayo.
Pharmacokinetics "tiapridal"
Maamulka muruqyada dhexdooda daroogada (200 mg) oo ay heerka ugu badnaan in jidhka la ogaado 30 daqiiqo ka dib, iyadoo la isticmaalayo kiniinka at dose isku mid ah - 60 daqiiqo. bioavailability ee daroogada isla markiiba marka loo isticmaalo cuntada ka hor 75% kor u kacay 95%. Maxaa yeelay, daawooyinka la isticmaalo kordhay sida iyo heerka ugu badnaan in u shaqeeyo ah (40%).
Nuugista ee jidhku waa gaabis ah in bukaanka dadka waayeelka ah. "Tiapridal" tilmaamaha loo isticmaalo waxaa loola jeedaa wakiil gudbaya caqabadaha mandheerta iyo dhiig-maskaxda. Waxaa la og yahay in inta lagu jiro daaweynta daroogada waxa ay joogtaa oo sideeda oo caanaha naaska. In haweenka, ka kaxayntu ay qayb ka mid ah daroogada ka dhaqso badan in ka mid ah ragga (in ka badan 2.9 saac), farqiga u yahay 0.7 saacadood. Dheef-lagu gartaa sida dhexdhexaad ah. Qaybta ugu muhiimsan ee daroogada (70%) laga saaro jidhka ka by kelyaha beddelin.
Tilmaamayaasha "Tiapridal" diyaarinta
Si loo fuliyo therapy la daroogada "Tiapridal" reading sida soo socota:
- Tardive (dyskinesia, lama filaan ah);
- Gilles de la Tourette Syndrom,
- chorea;
- xanuunada dabeecadda (state dagaal badan, cadhoodaan et al.), taasoo keentay in socodka la taaban karo ee Khamriga chronic iyo bukaanada waayeelka ah,
- daliilka xun ee dhaqanka, sida gobolka dagaal badan iyo caro;
- xanuun qof degdeg ah (foomka chronic).
Sababo, xadeynta si ay u helaan "Tiapridal" daroogada
Mamnuucayaa rogida tilmaamo "Tiapridal" loo isticmaalo carruurta da'doodu ka yar tahay lix sannadood. In daaweynta carruurta waa la fuliyay kiniini oo kaliya. Daawada waa in aan la daaweyn haweenka uurka leh iyo bukaan naas. Daawada looma isticmaalo in ay dhacdo diidmo in qaybaha, iyo siyaabo kale sida. Sababo ka mid ah wadamada sida:
- cagaarshowga iyo kelyaha, taas oo uu leeyahay darnaanta badan;
- prolaktinzavisimogo ogaado burooyinka, shaki ah ay joogaan,
- dhibaatooyinka hypertensive;
- ogaanshaha of pheochromocytoma, shaki ah jiritaankeeda.
Kiniiniyada iyo xal la wada isticmaalo "sultopride" iyo agonister receptor dopamine (marka laga reebo waa daaweynta bukaannada qaba cudurka Parkinson) ma weheliso qaar ka mid ah neuroleptics, wakiilada anti-arrhythmic ay leeyihiin fasalo aniga iyo III A.
Medicating "Tiapridal" edbinta ma ogola in isku mar la isticmaalayo "Moxifloxacin", "sparfloxacin", "Difemanila", "erythromycin", "bepridil," "mizolastine", "levodopa", "cisapride" iyo xididka "vincamine" .
Haddii bukaanka (gaar ahaan dadka waayeelka ah) Lagu daawaynayo daawo kuwaas oo keeni kara horumarinta hypokalemia, daraysa tabinta wadnaha, hagaagay bareeg QT, dhacdo ee bradycardia muujiyeen qof, isticmaal "Tiapridal" Waa in si taxadar leh. Digniin loo baahan yahay in kiisaska noocaas ah:
- cudurka Parkinson,
- lagu dhasho QT qof muruqa bareeg;
- hypokalemia;
- renal failure raaga,
- bradycardia;
- cudurada kuwaas oo khalkhal nidaamka wadnaha (tallaabo decompensation);
- qalalka.
Daaweynta la "Tiapridal"
on codsiga ah ee "Tiapridal" Buuggan ku talinaysaa in la isticmaalayo marka hore in yar ka qaataan, si tartiib ah iyaga kordhaya, si ay u helaan saamayn ugu badan.
xanuunada dabeecadda
Waayo, gargaarka waa loo baahan yahay si aad u dalbato 200 mg ah ee daawada maalin kasta (ilaa 300). Saamaynta wanaagsan waxaa lagu gaarayaa in lix isbuuc celcelis ahaan. bukaanka Older maamula qiyaas hoose ee daawada - 50 mg. dose A hal waa in la laba jeer baabbi'iyey maalin, iyo midhaha waa la ogol yahay in la raacayo bareeg u khaaska ah, tallaabada lagu sameeyaa si tartiib tartiib ah, iyada oo talo khabiir account. Qiyaasta maalin walba waa in aan ka badnayn 300 mg.
xanuun daran Chronic
dose maalin walba ah ee daroogada si loogu daweeyo xaaladaha sida waa ka 200 ilaa 400 mg.
Chorea, Gilles de la Tourette Syndrom
Marka fulinta daaweynta dose maalin kasta ilmahaaga la doorto iyada oo la tixgelinayo miisaanka jidhka oo ku saabsan 3-6 mg / kg. Haddii aad u baahan tahay si ay u qabtaan therapy qof weyn, marka hore loo isticmaalay 25 mg ah ee daawada maalin kasta, ka dib (ka dib markii korodh ah ee dose) - 300-800 mg.
Cadhoodaan, gardarada
Qiyaasta talinayaa maalin walba of medicament waa ka 100 ilaa 150 mg.
xanuunada dabeecadda
Qiyaasta talinayo in la isticmaalo maalintii (200 ilaa 300 mg) in ay dhacdo dalalka delirious ama predelirioznogo gaartay 400-1200 mg. Qiyaasta ugu badan ee suurtogalka ah taas waa in maaha in la dhaafo, waa 1800 mg. hordhaca ah ee daroogada soo saaray celcelis ahaan saacadood shan kasta. Haddii daawaynta lagama maarmaanka u ah qofka waayeelka ah, maalin walba waa 2-3 irbado u dhexeeya oo lagu arkay bareeg of 6 saacadood. Waayo, dawaynta dadka qaba sida talinayaa qaato maalin ah 200 ilaa 300 mg ah medicament waqti loo ogol yahay in ay soo galaan in ka yar 100 mg "tiapridal".
hadal xooggan ee dabiiciga ah ee joogtada ah ee xanuunka
Daaweynta ku salaysan qiyaasta ay maamusho maalin walba u dhiganta 200-400 mg ah ee daawada.
Dhibaatooyinka ay keento marka la qaadanayo "Tiapridal" daroogada
Marka daaweynta Buugga daroogada "Tiapridal" edbinta, dib u eegista xaqiijin suurtagalnimada dhibaato gaar ah. Ku xadgudubka ku dhici kara Fistula ah, neerfaha, hormoonada jidhka iyo nidaamka wadnaha iyo. Intaa waxaa dheer, waxaa jira halis of dhibaatooyin la xiriira dareenka. Waayo saamaynta taban kale waxaa ka mid ah xasaasiyad, daliilka maqaarka Ulasocto korodh miisaan, hypotension orthostatic.
Iska badinta "tiapridal"
Haddii aad isticmaasho dose xad-dhaaf ah badinta suurto gal ah iyo astaamaha ay ka mid rabshooyin miyir, ugu daran taasoo - kooma, syndrome neuroleptic (malignant, foomamka ba'an). Si aad u daaweyso xaaladda noocan ah u shaqeeyo waxaa lagu fuliyaa daaweynta ku salaysan wakiilada anticholinergic. Ka dib markii la baabiiyo of daroogada lagama maarmaan ah si ay u fuliyaan daaweyn astaamaha iyo plasmapheresis.
ganaaxyada
Ka hor inta isticmaalka daawada "Tiapridal" diiwaanka a ku talinaysaa in aad saxdo hypokalemia. Inta lagu guda jiro daawaynta waxaa muhiim ah in si joogto ah loola socdo dheelitirka elektrolytka, qaban-joogaha, ula socdaan isbedelka sawirka kiliinikada.
Haddii ay lagama maarmaan tahay in aad dalbato daroogada anticholinergic keeni helo neuroleptics syndrome extrapyramidal horumariyo halkii agonist receptor dopamine.
Waqtiga daaweynta waa in ay ka tanaasulaan howlaha in ay khatar ku iman karta, waxaa laguma talinayo in la sameeyo shaqo u baahan daryeel gaar ah iyo jawaab deg deg ah.
Dhexgalka waxyaabaha kale ee
diyaarinta isku darka qaar ka mid ah qaadashada daawooyinka "Tiapridal" edbinta, feedback la xiriira itimaalka ee dhacdo of falcelinta aan loo baahnayn. Waxaa laguma talinayo inta lagu jiro daaweynta codsatay "Clonidine", xasaasiyadda, anxiolytics, barbiturates iyo opioids, sida "tiapridal" saamayn doonaan fahmayaan. Sababo la incompatibility waa in aan loo qaadan "levodopa" iyo khamriga. Daawooyinka la isku dari karaa iyadoo la isticmaalayo neurotrophic daroogada, analgesics, murugada, neuroleptics. khatarta sare ee hypotension orthostatic, waxaa jira isticmaalka isku mar daroogada antihypertensive leh "Tiapridalom".
Qiimaha analogues daroogada, dib u ah oo ku saabsan daroogada "Tiapridal"
Haddii daaweynta lagama maarmaanka ah "Tiapridal" waxaa loola jeedaa description edbinta ha aad u ogaato wixii daroogadu waa. Qiimaha daroogada waa muhiimad weyn ee doorashada ee medicament ah si loogu soo daweeyo. Xalka in fijaan oo la iibsan karaa oo ku saabsan 995 rubles, iyo murriyado - for 1,400 rubles.
Waxaa ka mid ah analogues daroogada - "Eglonil", "Betamax". Of keydka laga yaabaa in lagu soo xulay "Sulpiride" ama "Prosulpin". Waxaa jira analoogga kale ee daroogada - "tiaprid", ayuu waxaa loo arkaa inta badan la heli karo, waa arrin ikhtiyaarka ah oo caan ah, soo-saarka daawada gudaha oo ka hadlaya shirkadda "Organic". Iyadoo qayb ka ah "tiaprid" bandhigaan walax isku mid ah oo firfircoon, taas oo ah qayb ka mid ah daawada "Tiapridal". analogs Isticmaalka Guide ku talinaysaa in ay doortaan, marka asalka ah isku mar ma loo isticmaali karaa daawooyinka qaar wuxuu sababaa waxyeelo iyo ma bixiso saamayn doonayo. Si daroogada ahaa ugu waxtarka badan, xisaabta badan oo dhibcood galay markii la doortay.
Inta lagu jiro daaweynta, waxaa muhiim ah in la raaco talo iyo talooyinka dhakhtarka oo dhan, taas oo ka kooban tilmaamaha loo isticmaalo. "Tiapridal", sida lagu muujiyey by-celin, in kiisaska intooda badan, waxaa loo isticmaalaa in la baabi'iyo xaaladaha weheliyay farax habdhiska iyo dhaqanka dagaalka ah, psychosis khamriga. Sida caadiga ah, bukaan iyo dhakhaatiirta ku qanacsanayn natiijada therapy. Asal ahaan, koorso kororsi looma baahna waayo sababta in saamayn la doonayo waxaa lagu soo koraya ka dib markii fulinta dabcan ugu horeysay. Reviews muujinaya in daawada bukaan "Tiapridal" fududahay in la isticmaalo.
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