CaafimaadkaDiyaarinta

"Tsinarin": tilmaamaha loo isticmaalo, dhigooda dhabta ah

blockers Calcium channel yeedhay group Nuurre Aw daroogada in ay leeyihiin mabda'a isku mid ah hawlgalka, laakiin ku kala duwan yihiin guryaha qaar ka mid ah, oo ay ku jirto ku soo koobin ogeed, selectivity nudaha iyo saamaynta on garaaca wadnaha.

mabda'a aasaasiga ah ee hawlgalka daawooyinka sida waa in ay awoodaan in ay la xakameeyo wax lays of udhigo Ca ka bannaan ee extracellular galay xididdada dhiigga iyo unugyada muruqa wadnaha via channels calcium (hakin) waa. Tani waxay keenaysaa in tallaabo vasodilator fahmayaan.

The ugu caansan antagonist calcium waa "tsinarin" daroogada. Tilmaamaha loogu isticmaalo, qiimaha, iyo dib u eegis kooban ee lacagta la hoos lagu qeexay doonaa.

foomka sii daayo, baakadaha, sharaxaad, halabuurka

Drug "tsinarin", dib u eegista ah kuwaas oo wanaagsan, waxaa suuq qaab biconvex, wareega iyo kiniinada cadcad. Waxa ay qayb weyn waa cinnarizine. waxa laga reebo, oo sideeda oo daroogada ka kooban yahay sida K25 excipients povidone, lactose, istaarijka sarreen, Silicon Kolloidol dioxide iyo milmahayn magnesium.

Taas macnaheedu waxa aad ka iibsan kartaa in unugyada dusha ka.

sifooyinka alaabta

arjiga ku of Guide "tsinarin" daroogada ayaa sheegay in antagonist xulashada of channels calcium (hakin). Waxay yaraynaysaa socodka Ca ra'iyi unugyada iyo yaraynaysaa tirada plasmolemma saldhig ah, laakiin sidoo kale kor u saamayn vasodilating ee carbon dioxide iyo yaraynaysaa cabirida xaalada muruqa ah arterioles ah.

By simaha si toos ah on weelashii, daroogada si weyn u yaraynaysaa ay jawaab u nafaqooyin (norepinephrine, epinephrine, angiotensin, Horomonka, iyo dopamine). Sidoo kale ogsoonow in medicament u tixgeliyo ayaa vasodilating guryaha, oo ay ku jirto ee loo geeysanayo maraakiibta cerebral. Xaaladdan oo kale, waxay leedahay saameyn ah kuma laha cadaadiska dhiigga.

Drug "tsinarin", qiimaha kaas oo hoos ku qoran, waxaa lagu dhexdhexaad ah kaga hadlay hawlaha antihistamine, waxay yaraynaysaa excitability ee hay'adaha vestibular iyo yaraynaysaa midab ah ee NS dabacsanaadaan. daroogada Tani wax ku ool ah u dhaqmo sidii kaafi hore cerebrovascular iyo chronic. Dadka qaba wareegga durugsan oo yaraada waxay hagaajinaysaa socodka dhiigga oo dhan unugyada iyo xubnaha. Sidoo kale waa hab lagu yareeyo nafwaayay dhiigga, waxay kordhisaa barti ee xuub ee unugyada dhiigga cas iyo iska caabin muruqa in hypoxia.

The kinetics daroogada

Waa maxay astaamaha ogeed soo jireenka ah ee daroogada "tsinarin"? Tilmaamaha Isticmaalka dhigayaa in wakiilka this waxaa resorbed ee mindhicirrada iyo caloosha. fiirsashada plasma sarreysey gaarey saddex saacadood ka dib. Isgaarsiinta la borotiinada plasma cinnarizine waa 91%. Daawada si buuxda loo metabolized beerka. Its wakhti badhkiis-nolosha waa afar saacadood. Waxaa soo baxday daawada ee kaadida iyo saxarada.

maragga

Drug "tsinarin" waxa muujiyay at dhaweynta:

  • dementia neefo;
  • stroke ischaemic;
  • xamilo cranial;
  • xaaladaha post-stroke (oo ay ku jiraan in stroke dhiigbaxa);
  • encephalopathy vascular,
  • waayo, kinetoses prophylaxis ah (badda ama cudur hawada, iyo sidoo kale inta lagu guda jiro ruxid);
  • xanuunada vestibular (oo ay ku jiraan la cudurka Meniere ee, tinnitus, vertigo, nystagmus, matag iyo lallabo asal labyrinthine);
  • xanuunka dhanjafka (ka hortagga weerarada);
  • xadgudub ku ah wareegga durugsan.

Sababo si ay u helaan Alwaaxdii

Under waxa xaaladaha waa in aan lagu soo qoray "tsinarin" daroogada? Tilmaamaha loogu isticmaalo warar sheegaya in daawaynta this waa u in:

  • diidmo,
  • wallaca;
  • naas-nuujinta.

Sidoo kale waa in la ogaadaa in daawada la qoray si taxadir leh in cudurka Parkinson.

Drug "tsinarin": tilmaamaha loo isticmaalo

kiniiniyada Qaadashada waa in loo arko gudaha, doorbidayaa cuntada ka dib.

Marka dhibtay, daawo wareegga dhiigga maskaxda maamusho qadarkuu of 25-50 mg saddex jeer maalintii, iyo wareegga dhiigga durugsan - at 50-75 mg la badnaanta isku.

Marka xanuunada vestibular talinayaa in ay qaataan daawada at 25 mg saddex jeer maalintii. Marka kinetosis ama waxa loogu yeero "wadada" bukaanka cudurka dadka waaweyn ay maamusho 25 mg daroogada 30 daqiiqo safarka ka hor. Haddii loo baahan yahay, daawada qaato soo noqnoqda 6 saacadood ka dib (ee lacagta la mid ah).

Waayo, carruurta, daroogada taas waxaa loo qoray in xaddiga 1/2 of qiyaasta dadka waaweyn ah.

At dareen sare si ay therapy ah medicament bilaabmaa qiyaasta qeybtii tartiib ah u kordhi. koorsada daawada socon karaa meel kasta oo ka 2-3 todobaad ilaa dhawr bilood.

waxyeellooyin

daroogada Tani waxay keeni kartaa soo socda reactions dhinaca:

  • afka oo qalala, dyspepsia, xanuun gaastari, joonis cholestatic;
  • hurdo, madax xanuun, daal, iyo disorder extrapyramidal (tusaale ahaan, kor u cabirida xaalada muruqa, gariirka ee addimada, hypokinesia);
  • lichen planus ', dhidid, lupus-sida syndrome, finan maqaarka ah,
  • saamaynta xasaasiyad, miisaanka oo kordha, hoos u cadaadiska dhiigga.

Price, fasax analogues daroogada iyo dib u eegis ku saabsan

-Bixinta daawooyinka ka tirsan kooxda reer blockers calcium channel, qaadeen by warqad dhakhtar. Price of daroogada ku saabsan tahay 20-50 rubles.

Haddii loo baahdo, qalabka lagu beddeli karo daroogada "Vertizin", "Diziron", "Stugezin", "stugeron", "Tsinazin", "Tsinedil" "Cinnarizine" iyo si bixi.

macaamiisha Inta badan qaadato antagonist this, ku doodaya in ay tahay maandooriye aad u hufan oo wax ku ool ah. Kiniinka "tsinarin" caawisaa baabi'iyo xanuunada vestibular iyo cudura ee geedi socodka wareegga dhiigga. Intaa waxaa dheer, daroogada uu leeyahay saamayn togan ku jidhka bini'aadamka la jaf, neefo dementia iyo xaaladaha post-stroke.

Sidoo kale waa in Waxaan la soco in wakiilka loo arkaa inta badan sababa falcelinta kooxda. Si looga hortago horumarinta, waa in si adag u hoggaansamaan dhammaan talooyinka dhakhtarka. Qaado pill "tsinarin" ee ikhtiyaarka kaliya, Waxaa reebban. Waa in loo qoro oo kaliya uu dhakhtarka xaadirka ah.

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